Category: Reagents

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Reference: 29073-25

An active ginsenoside metabolite; cytotoxic to HL-60 cancer cells (IC50 = 16 µM); inhibits the proliferation of HUVECs (EC50 = 6.64 µg/ml); blocks LPS-induced increases in the protein levels of COX-2 and iNOS and decreases LPS-induced NF-κB activity in RAW 264.7 cells from 1-20 µM

Reference: 18619-250

An adrenergic α1A receptor agonist (Ki = 1.4 µM) that demonstrates selectivity against the α1B and α1C receptor subtypes (Kis = 23.9 and 47.8 µM, respectively); frequently used to precontract smooth muscle in preparations designed to study the properties of various vasodilator agents

Reference: B5701-50

sphingosine-1-phosphate receptor 1 (S1P1) agonist

Reference: 29073-5

An active ginsenoside metabolite; cytotoxic to HL-60 cancer cells (IC50 = 16 µM); inhibits the proliferation of HUVECs (EC50 = 6.64 µg/ml); blocks LPS-induced increases in the protein levels of COX-2 and iNOS and decreases LPS-induced NF-κB activity in RAW 264.7 cells from 1-20 µM

Reference: 18619-50

An adrenergic α1A receptor agonist (Ki = 1.4 µM) that demonstrates selectivity against the α1B and α1C receptor subtypes (Kis = 23.9 and 47.8 µM, respectively); frequently used to precontract smooth muscle in preparations designed to study the properties of various vasodilator agents

Reference: B5702-5

Apelin receptor (APJ) antagonist

Reference: 29134-1

A form of Gb4 lacking the fatty acyl group; binds to VTE in a glycolipid binding assay; acylated to stearic acid via a condensation reaction by sphingolipid ceramide N-deacylase to form a ceramide

Reference: 18619-500

An adrenergic α1A receptor agonist (Ki = 1.4 µM) that demonstrates selectivity against the α1B and α1C receptor subtypes (Kis = 23.9 and 47.8 µM, respectively); frequently used to precontract smooth muscle in preparations designed to study the properties of various vasodilator agents

Reference: B5702-10

Apelin receptor (APJ) antagonist

Reference: 29176-1

A synthetic bile acid and a derivative of cholic acid; increases bile flow by 2.7-fold and decreases biliary levels of phospholipids, cholesterol, and bilirubin in conscious dogs at 50 mg/kg; increases bile flow by 253% at 1 µmol/min/0.1 kg and decreases the secretion rate of phospholipids and cholesterol by 64 and 94%, respectively, in rats when infused intravenously at 2 µmol/min/0.1 kg

Reference: 18622-1

A selective agonist of β3-adrenergic receptors with Ki values of 0.43, 9.17, and 37.9 µM for β3, β2, and β1, respectively

Reference: B5702-25

Apelin receptor (APJ) antagonist