Category: Reagents

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Reference: 19760-1

A potent CYP3A4 inhibitor (IC50s = 0.30 ppm in a cell-free assay, 0.33 µM in HL7 human liver cells, and 0.22 µM in S9 human intestine cells); inhibits the transport of talinolol, a P-gp/ABCB1 transporter substrate, across Caco-2 cell monolayers (IC50 = 0.7 µM); has insecticidal properties (5 µg/cm2 leads to 100% mortality of adult olive fruit flies)

Reference: 10007126-100

A synthetic intermediate useful for pharmaceutical synthesis

Reference: A2610-5.1

For pinworm treatment in animals

Reference: 19760-10

A potent CYP3A4 inhibitor (IC50s = 0.30 ppm in a cell-free assay, 0.33 µM in HL7 human liver cells, and 0.22 µM in S9 human intestine cells); inhibits the transport of talinolol, a P-gp/ABCB1 transporter substrate, across Caco-2 cell monolayers (IC50 = 0.7 µM); has insecticidal properties (5 µg/cm2 leads to 100% mortality of adult olive fruit flies)

Reference: 10007126-500

A synthetic intermediate useful for pharmaceutical synthesis

Reference: A2610-500

For pinworm treatment in animals

Reference: 19760-25

A potent CYP3A4 inhibitor (IC50s = 0.30 ppm in a cell-free assay, 0.33 µM in HL7 human liver cells, and 0.22 µM in S9 human intestine cells); inhibits the transport of talinolol, a P-gp/ABCB1 transporter substrate, across Caco-2 cell monolayers (IC50 = 0.7 µM); has insecticidal properties (5 µg/cm2 leads to 100% mortality of adult olive fruit flies)

Reference: A2612-S

Potent reversible proteasome inhibitor