Reagents (2)

10'-Desmethoxystreptonigrin

Reference: 28065-2,5

€0.00 (tax incl.)

An antibiotic; active against a variety of bacteria, including S. aureus, S. faecalis, E. coli, K. pneumoniae, and P. vulgaris (MICs = 0.4, 1.6, 3.1, 3.1, and 0.4 µg/ml, respectively); cytotoxic to HCT116 colon and...

Neoaureothin

Reference: 28091-2,5

€0.00 (tax incl.)

A bacterial metabolite; an AR antagonist that inhibits binding of DHT to ARs (IC50 = 13 μM); inhibits DHT-induced expression of prostate-specific antigen in LNCaP cells (IC50 = 1.75 nM); is cytotoxic to A549, HCT116,...

SCH 38519

Reference: 28092-2,5

€0.00 (tax incl.)

A fungal metabolite; inhibits thrombin-induced aggregation, as well as inhibits serotonin secretion in human platelets (IC50s = 68 and 61 µg/ml, respectively); inhibits the growth of various Gram-negative and...

Saccharocarcin A

Reference: 28094-2,5

€0.00 (tax incl.)

An antibiotic; active against M. luteus, S. aureus, E. coli, P. aeruginosa, and C. albicans in a disc assay; inhibits C. trachomatis infection in McCoy cells,,

Nybomycin

Reference: 28099-2,5

€0.00 (tax incl.)

A fungal metabolite with antibacterial activity; active against B. subtilis, B. cereus, B. mycoides, M. smegmatis, and K. pneumoniae (MICs = 0.025, 2, 0.8, 0.2, and 0.003 μg/ml, respectively); active against M....

1-Alaninechlamydocin

Reference: 28102-2,5

€0.00 (tax incl.)

An HDAC inhibitor; reduces total HDAC activity in HeLa cell lysates; reduces proliferation of MIA PaCa-2, PANC-1, and hTERT-HPNE cells (GI50s = 5.3, 14, and 2.0 nM, respectively)

TAN 420E

Reference: 28120-2,5

€0.00 (tax incl.)

A bacterial metabolite; scavenges DPPH radicals in vitro (IC50 = 1.3 μM); reduces TBARS in rat liver microsomes by 72% at 100 μg/ml; is active against B. brevis, B. cereus, M. flavus, and S. aureus (MICs = 50-100...

Geninthiocin A

Reference: 28125-2,5

€0.00 (tax incl.)

A cyclic thiopeptide bacterial metabolite; active against a variety of Gram-positive bacteria (MICs = 0.2-4 µg/ml), the Gram-negative bacterium C. violaceum (MIC = 19 µg/ml), and the fungus M. hiemalis (MIC = 38...

Avenaciolide

Reference: 28128-2,5

€0.00 (tax incl.)

A fungal metabolite; inhibits glutamate transport in isolated rat liver mitochondria (Ki = 8 μM)

Desotamide

Reference: 28129-2,5

€0.00 (tax incl.)

A cyclic hexapeptide antibiotic; active against S. aureus, S. pneumoniae, and MRSE (MICs = 16, 12.5, and 32 μg/ml, respectively)

Decatromicin B

Reference: 28132-2,5

€0.00 (tax incl.)

A bacterial metabolite; active against Gram-positive bacteria, including several strains of S. aureus (MICs = 0.39-0.78 µg/ml), two strains of MRSA (MICs = 0.39 and 0.78 µg/ml), as well as M. luteus, B. subtilis, and...

Sporidesmolide II

Reference: 28133-2,5

€0.00 (tax incl.)

A cyclic depsipeptide,

Telomycin

Reference: 28137-2,5

€0.00 (tax incl.)

A macrocyclic peptide lactone antibiotic; active against Gram-positive bacteria, including S. aureus, MRSA, and E. faecium (MICs = 4, 2, and 16 µg/ml, respectively); eradicates B. anserina spirochetosis infection in...

Quinaldopeptin

Reference: 28167-2,5

€0.00 (tax incl.)

A quinomycin antibiotic; active against a variety of bacteria, including S. pyogenes, S. aureus, C. perfringens, S. faecalis, E. coli, and K. pneumoniae (MICs = 0.2, 0.4, 0.8, 1.6, 3.1, and 6.3 µg/ml, respectively);...

Leucinostatin A

Reference: 28190-2,5

€0.00 (tax incl.)

A fungal metabolite with diverse biological activities; active against various fungi and bacteria in a disc assay; reduces TPA- and anti-CD3 antibody-induced T cell activation from 0.1-1 μg/ml; inhibits proliferation...

Methylspinazarin

Reference: 29898-2,5

€0.00 (tax incl.)

A bacterial metabolite and COMT inhibitor (IC50 = 0.8 μg/ml); selective for COMT over tyrosine hydroxylase, DOPA decarboxylase, and dopamine-β-hydroxylase at 100 μg/ml; decreases blood pressure in spontaneously...

Polygodial pyridazine

Reference: 29900-2,5

€0.00 (tax incl.)

A derivative of polygodial; inhibits the growth of MCF-7 and Hs 683 cells (GI50s = 72 and 93 μM, respectively)

Byssochlamic Acid

Reference: 29908-2,5

€0.00 (tax incl.)

A mycotoxin; lethal to mice (LD50 = 94 mg/kg)

Aszonapyrone A

Reference: 29940-2,5

€0.00 (tax incl.)

A meroditerpene fungal metabolite with diverse biological activities; inhibits the growth of MCF-7, NCI H460, and A375-C5 cancer cells (GI50s = 13.6, 11.6, and 10.2 μM, respectively); active against...

Territrem A

Reference: 29941-2,5

€0.00 (tax incl.)

A mycotoxin originally isolated from A. terreus; irreversibly inhibits AChE (IC50 = 24 nM for the electric eel enzyme); induces tremors in mice with a median tremulous dose of 0.31 mg/kg; LD50 = 17.6 mg/kg

Monomethylsulochrin

Reference: 29942-2,5

€0.00 (tax incl.)

A fungal metabolite; active against H. pylori (MIC = 10 µg/ml)

Chevalone E

Reference: 29948-2,5

€0.00 (tax incl.)

A meroterpene; has been found in A. similanensis

Novobiocic Acid

Reference: 29966-2,5

€0.00 (tax incl.)

An aglycone form of novobiocin

Asperfuran

Reference: 29989-2,5

€0.00 (tax incl.)

A fungal metabolite; inhibits the growth of 23 fungi in a disc assay at 50 µg per disc; inhibits chitin synthase (IC50 = 300 µM); inhibits proliferation of HeLa S3 and L1210 cancer cells (IC50s = 25 µg/ml for both)

(–)-Himgaline

Reference: 29990-2,5

€0.00 (tax incl.)

An alkaloid; has been found in G. belgraveana

Himandridine

Reference: 30055-2,5

€0.00 (tax incl.)

An alkaloid

Himbosine

Reference: 30056-2,5

€0.00 (tax incl.)

An alkaloid; has been found in H. baccata bark

Janthitrem A

Reference: 30166-2,5

€0.00 (tax incl.)

A mycotoxin; induces tremors in mice and decreases the time to fall from the rotarod at 4 mg/kg; reduces W. cervinata larvae weight gain and food consumption at 20 µg/g

Pikromycin

Reference: 31331-2,5

€0.00 (tax incl.)

A macrolide antibiotic; active against E. coli, S. aureus, and B. subtilis (MIC99s = 50-60, 90-100, and 25-30 µM, respectively)

Beauveriolide III

Reference: 31775-2,5

€0.00 (tax incl.)

A cyclodepsipeptide inhibitor of lipid droplet formation; inhibits lipid droplet formation at 3 and 10 µM and inhibits cholesterol synthesis (IC50 = 0.41 µM) in primary mouse peritoneal macrophages; inhibits ACAT...

Amicoumacin B

Reference: 31777-2,5

€0.00 (tax incl.)

An amicoumacin with quorum-sensing inhibitory activity; active against C. violaceum (MIC = 250 µg/ml); increases the expression of BMP2 in MG-63 cells

S-5751

Reference: 10004030-1

€0.00 (tax incl.)

A selective antagonist of DP1 (Ki = 1.6 nM); blocks PGD2-induced plasma exudation in the conjunctiva (ED50 = 0.099 mg/kg) and suppresses antigen-induced allergic responses in guinea pigs

S-5751

Reference: 10004030-5

€0.00 (tax incl.)

A selective antagonist of DP1 (Ki = 1.6 nM); blocks PGD2-induced plasma exudation in the conjunctiva (ED50 = 0.099 mg/kg) and suppresses antigen-induced allergic responses in guinea pigs

S-5751

Reference: 10004030-500

€0.00 (tax incl.)

A selective antagonist of DP1 (Ki = 1.6 nM); blocks PGD2-induced plasma exudation in the conjunctiva (ED50 = 0.099 mg/kg) and suppresses antigen-induced allergic responses in guinea pigs

Luteolin

Reference: 10004161-10

€0.00 (tax incl.)

A potent flavanoid inhibitor of soybean and reticulocyte 15-LOs (IC50 = 0.6 µM)

Luteolin

Reference: 10004161-100

€0.00 (tax incl.)

A potent flavanoid inhibitor of soybean and reticulocyte 15-LOs (IC50 = 0.6 µM)

Luteolin

Reference: 10004161-50

€0.00 (tax incl.)

A potent flavanoid inhibitor of soybean and reticulocyte 15-LOs (IC50 = 0.6 µM)

Luteolin

Reference: 10004161-500

€0.00 (tax incl.)

A potent flavanoid inhibitor of soybean and reticulocyte 15-LOs (IC50 = 0.6 µM)

Apoptosis Activator 2

Reference: 10004176-10

€0.00 (tax incl.)

Promotes the cytochrome c-dependent oligomerization of Apaf-1 into the mature apoptosome, thus increasing procaspase-9 processing and subsequent caspase-3 activation; induces apoptosis in leukemia cells (IC50 = 4-9 μM)

Apoptosis Activator 2

Reference: 10004176-25

€0.00 (tax incl.)

Promotes the cytochrome c-dependent oligomerization of Apaf-1 into the mature apoptosome, thus increasing procaspase-9 processing and subsequent caspase-3 activation; induces apoptosis in leukemia cells (IC50 = 4-9 μM)

Apoptosis Activator 2

Reference: 10004176-5

€0.00 (tax incl.)

Promotes the cytochrome c-dependent oligomerization of Apaf-1 into the mature apoptosome, thus increasing procaspase-9 processing and subsequent caspase-3 activation; induces apoptosis in leukemia cells (IC50 = 4-9 μM)

Apoptosis Activator 2

Reference: 10004176-50

€0.00 (tax incl.)

Promotes the cytochrome c-dependent oligomerization of Apaf-1 into the mature apoptosome, thus increasing procaspase-9 processing and subsequent caspase-3 activation; induces apoptosis in leukemia cells (IC50 = 4-9 μM)

CAY10443

Reference: 10004177-10

€0.00 (tax incl.)

A pro-apoptotic activator of the apoptosome; activates caspase-3 (EC50 = 5 µM) in a cell free, multi-component assay,

CAY10443

Reference: 10004177-25

€0.00 (tax incl.)

A pro-apoptotic activator of the apoptosome; activates caspase-3 (EC50 = 5 µM) in a cell free, multi-component assay,

CAY10443

Reference: 10004177-5

€0.00 (tax incl.)

A pro-apoptotic activator of the apoptosome; activates caspase-3 (EC50 = 5 µM) in a cell free, multi-component assay,

CAY10443

Reference: 10004177-50

€0.00 (tax incl.)

A pro-apoptotic activator of the apoptosome; activates caspase-3 (EC50 = 5 µM) in a cell free, multi-component assay,

NESS 0327

Reference: 10004184-1

€0.00 (tax incl.)

An extremely potent cannabinoid receptor antagonist with high selectivity for the central CB1 receptor (Ki = 0.35 pM) compared to the peripheral CB2 receptor (Ki = 21 nM)

NESS 0327

Reference: 10004184-10

€0.00 (tax incl.)

An extremely potent cannabinoid receptor antagonist with high selectivity for the central CB1 receptor (Ki = 0.35 pM) compared to the peripheral CB2 receptor (Ki = 21 nM)

NESS 0327

Reference: 10004184-5

€0.00 (tax incl.)

An extremely potent cannabinoid receptor antagonist with high selectivity for the central CB1 receptor (Ki = 0.35 pM) compared to the peripheral CB2 receptor (Ki = 21 nM)

3,4',5-Trismethoxybenzophenone

Reference: 10004185-10

€0.00 (tax incl.)

An analog of trimethoxy resveratrol; inhibits the growth of a variety of human tumor cell lines at concentrations form 0.4 to 2 µg/ml, which is 5-6 times more potent than resveratrol

3,4',5-Trismethoxybenzophenone

Reference: 10004185-100

€0.00 (tax incl.)

An analog of trimethoxy resveratrol; inhibits the growth of a variety of human tumor cell lines at concentrations form 0.4 to 2 µg/ml, which is 5-6 times more potent than resveratrol

3,4',5-Trismethoxybenzophenone

Reference: 10004185-25

€0.00 (tax incl.)

An analog of trimethoxy resveratrol; inhibits the growth of a variety of human tumor cell lines at concentrations form 0.4 to 2 µg/ml, which is 5-6 times more potent than resveratrol

3,4',5-Trismethoxybenzophenone

Reference: 10004185-50

€0.00 (tax incl.)

An analog of trimethoxy resveratrol; inhibits the growth of a variety of human tumor cell lines at concentrations form 0.4 to 2 µg/ml, which is 5-6 times more potent than resveratrol

(S)-Flurbiprofen

Reference: 10004207-1

€0.00 (tax incl.)

The COX-active enantiomer of flurbiprofen (IC50s = 0.48 and 0.47 µM for COX-1 and COX-2, respectively); inhibits the release of 6-keto-PGF1α and TXB2 from rat whole blood, gastric mucosa, lung, and jejunal tissue ex...

(S)-Flurbiprofen

Reference: 10004207-100

€0.00 (tax incl.)

The COX-active enantiomer of flurbiprofen (IC50s = 0.48 and 0.47 µM for COX-1 and COX-2, respectively); inhibits the release of 6-keto-PGF1α and TXB2 from rat whole blood, gastric mucosa, lung, and jejunal tissue ex...

(S)-Flurbiprofen

Reference: 10004207-250

€0.00 (tax incl.)

The COX-active enantiomer of flurbiprofen (IC50s = 0.48 and 0.47 µM for COX-1 and COX-2, respectively); inhibits the release of 6-keto-PGF1α and TXB2 from rat whole blood, gastric mucosa, lung, and jejunal tissue ex...

(S)-Flurbiprofen

Reference: 10004207-500

€0.00 (tax incl.)

The COX-active enantiomer of flurbiprofen (IC50s = 0.48 and 0.47 µM for COX-1 and COX-2, respectively); inhibits the release of 6-keto-PGF1α and TXB2 from rat whole blood, gastric mucosa, lung, and jejunal tissue ex...

SC-236

Reference: 10004219-1

€0.00 (tax incl.)

A potent, selective, orally active inhibitor of COX-2 with an IC50 value of 10 nM and approximately 18,000-fold selectivity for COX-2 over COX-1

SC-236

Reference: 10004219-10

€0.00 (tax incl.)

A potent, selective, orally active inhibitor of COX-2 with an IC50 value of 10 nM and approximately 18,000-fold selectivity for COX-2 over COX-1

SC-236

Reference: 10004219-5

€0.00 (tax incl.)

A potent, selective, orally active inhibitor of COX-2 with an IC50 value of 10 nM and approximately 18,000-fold selectivity for COX-2 over COX-1

SC-236

Reference: 10004219-50

€0.00 (tax incl.)

A potent, selective, orally active inhibitor of COX-2 with an IC50 value of 10 nM and approximately 18,000-fold selectivity for COX-2 over COX-1

cis-Resveratrol

Reference: 10004235-10

€0.00 (tax incl.)

Double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers; exhibits antioxidant activity in the micromolar range similar to that observed with trans-resveratrol

cis-Resveratrol

Reference: 10004235-100

€0.00 (tax incl.)

Double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers; exhibits antioxidant activity in the micromolar range similar to that observed with trans-resveratrol

cis-Resveratrol

Reference: 10004235-5

€0.00 (tax incl.)

Double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers; exhibits antioxidant activity in the micromolar range similar to that observed with trans-resveratrol

cis-Resveratrol

Reference: 10004235-50

€0.00 (tax incl.)

Double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers; exhibits antioxidant activity in the micromolar range similar to that observed with trans-resveratrol

Abnormal Cannabidiol

Reference: 10004259-1

€0.00 (tax incl.)

An agonist of GPR55 (EC50 = 2.5 µM in a GTPγS binding assay); selective for GPR55 over CB1 and CB2 (EC50s = >30 µM for both in GTPγS binding assays); a full agonist at GPR18 (EC50 = 0.835 µM for inducing p44/42 MAPK...

Abnormal Cannabidiol

Reference: 10004259-10

€0.00 (tax incl.)

An agonist of GPR55 (EC50 = 2.5 µM in a GTPγS binding assay); selective for GPR55 over CB1 and CB2 (EC50s = >30 µM for both in GTPγS binding assays); a full agonist at GPR18 (EC50 = 0.835 µM for inducing p44/42 MAPK...

Abnormal Cannabidiol

Reference: 10004259-25

€0.00 (tax incl.)

An agonist of GPR55 (EC50 = 2.5 µM in a GTPγS binding assay); selective for GPR55 over CB1 and CB2 (EC50s = >30 µM for both in GTPγS binding assays); a full agonist at GPR18 (EC50 = 0.835 µM for inducing p44/42 MAPK...

Abnormal Cannabidiol

Reference: 10004259-5

€0.00 (tax incl.)

An agonist of GPR55 (EC50 = 2.5 µM in a GTPγS binding assay); selective for GPR55 over CB1 and CB2 (EC50s = >30 µM for both in GTPγS binding assays); a full agonist at GPR18 (EC50 = 0.835 µM for inducing p44/42 MAPK...

GW 501516

Reference: 10004272-1

€0.00 (tax incl.)

PPARδ stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity. GW 501516 is the first highly selective synthetic PPARδ agonist...

GW 501516

Reference: 10004272-10

€0.00 (tax incl.)

PPARδ stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity. GW 501516 is the first highly selective synthetic PPARδ agonist...

GW 501516

Reference: 10004272-5

€0.00 (tax incl.)

PPARδ stimulation or over-expression in adipocytes leads to increased fatty acid oxidation, improved exercise tolerance, and resistance to obesity. GW 501516 is the first highly selective synthetic PPARδ agonist...

(±)-Nutlin-3

Reference: 10004372-1

€0.00 (tax incl.)

An inhibitor of p53-Mdm2 interaction (IC50 = 0.09 µM); induces the expression of p53-regulated genes and exhibits potent antiproliferative activity in cells with functional p53

(±)-Nutlin-3

Reference: 10004372-10

€0.00 (tax incl.)

An inhibitor of p53-Mdm2 interaction (IC50 = 0.09 µM); induces the expression of p53-regulated genes and exhibits potent antiproliferative activity in cells with functional p53

(±)-Nutlin-3

Reference: 10004372-5

€0.00 (tax incl.)

An inhibitor of p53-Mdm2 interaction (IC50 = 0.09 µM); induces the expression of p53-regulated genes and exhibits potent antiproliferative activity in cells with functional p53

(±)-Nutlin-3

Reference: 10004372-50

€0.00 (tax incl.)

An inhibitor of p53-Mdm2 interaction (IC50 = 0.09 µM); induces the expression of p53-regulated genes and exhibits potent antiproliferative activity in cells with functional p53

Sulindac

Reference: 10004386-1

€0.00 (tax incl.)

A non-selective inhibitor of both COX-1 and COX-2 with extensive epidemiology documenting its effective reduction of human colorectal cancer

Sulindac

Reference: 10004386-10

€0.00 (tax incl.)

A non-selective inhibitor of both COX-1 and COX-2 with extensive epidemiology documenting its effective reduction of human colorectal cancer

Sulindac

Reference: 10004386-5

€0.00 (tax incl.)

A non-selective inhibitor of both COX-1 and COX-2 with extensive epidemiology documenting its effective reduction of human colorectal cancer

Sulindac

Reference: 10004386-50

€0.00 (tax incl.)

A non-selective inhibitor of both COX-1 and COX-2 with extensive epidemiology documenting its effective reduction of human colorectal cancer

Sulindac sulfide

Reference: 10004387-1

€0.00 (tax incl.)

A metabolite of sulindac that inhibits both COX-1 and COX-2 (IC50s = 1.9 and 1.21 µM, respectively); also inhibits aldose reductase (IC50 = 279 nM), blocking NADPH-dependent reduction of glucose to sorbitol, and...

Sulindac sulfide

Reference: 10004387-10

€0.00 (tax incl.)

A metabolite of sulindac that inhibits both COX-1 and COX-2 (IC50s = 1.9 and 1.21 µM, respectively); also inhibits aldose reductase (IC50 = 279 nM), blocking NADPH-dependent reduction of glucose to sorbitol, and...

Sulindac sulfide

Reference: 10004387-25

€0.00 (tax incl.)

A metabolite of sulindac that inhibits both COX-1 and COX-2 (IC50s = 1.9 and 1.21 µM, respectively); also inhibits aldose reductase (IC50 = 279 nM), blocking NADPH-dependent reduction of glucose to sorbitol, and...

Sulindac sulfide

Reference: 10004387-5

€0.00 (tax incl.)

A metabolite of sulindac that inhibits both COX-1 and COX-2 (IC50s = 1.9 and 1.21 µM, respectively); also inhibits aldose reductase (IC50 = 279 nM), blocking NADPH-dependent reduction of glucose to sorbitol, and...

Reversine

Reference: 10004412-1

€0.00 (tax incl.)

A purine derivative; induces differentiation or dedifferentiation, depending on cell type; inhibits the Aurora A, B, and C kinases with IC50 values of 98-876 nM; A3 receptor antagonist (Ki = 0.66 µM); inhibits MPS1...

Reversine

Reference: 10004412-10

€0.00 (tax incl.)

A purine derivative; induces differentiation or dedifferentiation, depending on cell type; inhibits the Aurora A, B, and C kinases with IC50 values of 98-876 nM; A3 receptor antagonist (Ki = 0.66 µM); inhibits MPS1...

Reversine

Reference: 10004412-25

€0.00 (tax incl.)

A purine derivative; induces differentiation or dedifferentiation, depending on cell type; inhibits the Aurora A, B, and C kinases with IC50 values of 98-876 nM; A3 receptor antagonist (Ki = 0.66 µM); inhibits MPS1...

Reversine

Reference: 10004412-5

€0.00 (tax incl.)

A purine derivative; induces differentiation or dedifferentiation, depending on cell type; inhibits the Aurora A, B, and C kinases with IC50 values of 98-876 nM; A3 receptor antagonist (Ki = 0.66 µM); inhibits MPS1...

NADP+ (sodium salt hydrate)

Reference: 10004675-1

€0.00 (tax incl.)

The oxidized form of NADPH; serves as a cofactor in various biological reactions

NADP+ (sodium salt hydrate)

Reference: 10004675-100

€0.00 (tax incl.)

The oxidized form of NADPH; serves as a cofactor in various biological reactions

NADP+ (sodium salt hydrate)

Reference: 10004675-250

€0.00 (tax incl.)

The oxidized form of NADPH; serves as a cofactor in various biological reactions

NADP+ (sodium salt hydrate)

Reference: 10004675-50

€0.00 (tax incl.)

The oxidized form of NADPH; serves as a cofactor in various biological reactions

FMOC-L-Leucine

Reference: 10004888-100

€0.00 (tax incl.)

A partial agonist of PPARγ; activates PPARγ with a lower potency (Ki = 15 versus 0.035 µM) but a similar maximal efficacy compared to rosiglitazone; improves insulin resistance in normal, diet-induced...

FMOC-L-Leucine

Reference: 10004888-25

€0.00 (tax incl.)

A partial agonist of PPARγ; activates PPARγ with a lower potency (Ki = 15 versus 0.035 µM) but a similar maximal efficacy compared to rosiglitazone; improves insulin resistance in normal, diet-induced...

FMOC-L-Leucine

Reference: 10004888-50

€0.00 (tax incl.)

A partial agonist of PPARγ; activates PPARγ with a lower potency (Ki = 15 versus 0.035 µM) but a similar maximal efficacy compared to rosiglitazone; improves insulin resistance in normal, diet-induced...

O-1918

Reference: 10004914-1

€0.00 (tax incl.)

A cannabidiol (CBD) analog that acts as a selective antagonist of abnormal CBD (Abn-CBD) at the non-CB1/CB2 endothelial receptor; does not bind to CB1 or CB2 receptors at concentrations up to 30 µM and inhibits the...

O-1918

Reference: 10004914-10

€0.00 (tax incl.)

A cannabidiol (CBD) analog that acts as a selective antagonist of abnormal CBD (Abn-CBD) at the non-CB1/CB2 endothelial receptor; does not bind to CB1 or CB2 receptors at concentrations up to 30 µM and inhibits the...

O-1918

Reference: 10004914-25

€0.00 (tax incl.)

A cannabidiol (CBD) analog that acts as a selective antagonist of abnormal CBD (Abn-CBD) at the non-CB1/CB2 endothelial receptor; does not bind to CB1 or CB2 receptors at concentrations up to 30 µM and inhibits the...

O-1918

Reference: 10004914-5

€0.00 (tax incl.)

A cannabidiol (CBD) analog that acts as a selective antagonist of abnormal CBD (Abn-CBD) at the non-CB1/CB2 endothelial receptor; does not bind to CB1 or CB2 receptors at concentrations up to 30 µM and inhibits the...

N,N'-Dicyclohexylurea

Reference: 10004971-10

€0.00 (tax incl.)

A selective sEH inhibitor with IC50 values of 160 and 90 nM for recombinant human and mouse sEH, respectively; at 10 µM, blocks the hydrolysis of cis- and trans-EETs and completely inhibits 14,(15)-EET-induced PPAR...

Category: Reagents

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