Category: Reagents

Reference: 10004974-25
€0.00 (tax incl.)
A selective calcium ionophore that mobilizes intracellular calcium stores. It is used as a research tool to raise the intracellular level of calcium, to study calcium transport across biological membranes, and to...
Reference: 10004974-5
€0.00 (tax incl.)
A selective calcium ionophore that mobilizes intracellular calcium stores. It is used as a research tool to raise the intracellular level of calcium, to study calcium transport across biological membranes, and to...
Reference: 10004976-10
€0.00 (tax incl.)
A potent anti-fungal antibiotic that can directly block nuclear transport by inhibiting the action of CRM1
Reference: 10004976-25
€0.00 (tax incl.)
A potent anti-fungal antibiotic that can directly block nuclear transport by inhibiting the action of CRM1
Reference: 10004976-5
€0.00 (tax incl.)
A potent anti-fungal antibiotic that can directly block nuclear transport by inhibiting the action of CRM1
Reference: 10004985-1
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~7 µM); promotes the growth of HCT-116 cells ~20% at concentrations at or below 1 µM
Reference: 10004985-10
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~7 µM); promotes the growth of HCT-116 cells ~20% at concentrations at or below 1 µM
Reference: 10004985-5
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~7 µM); promotes the growth of HCT-116 cells ~20% at concentrations at or below 1 µM
Reference: 10005002-1
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~8 µM); promotes the growth of HCT116 cells ~40% at concentrations between 5-100 nM
Reference: 10005002-10
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~8 µM); promotes the growth of HCT116 cells ~40% at concentrations between 5-100 nM
Reference: 10005002-5
€0.00 (tax incl.)
A nutlin-3 analog; inhibits the growth of HCT116 cells at high concentrations (IC50 = ~8 µM); promotes the growth of HCT116 cells ~40% at concentrations between 5-100 nM
Reference: 10005019-1
€0.00 (tax incl.)
An HDAC inhibitor with an IC50 value of 30 µM when tested in HeLa cell nuclear extracts using 200 µM acetylated fluorometric substrate
Reference: 10005019-10
€0.00 (tax incl.)
An HDAC inhibitor with an IC50 value of 30 µM when tested in HeLa cell nuclear extracts using 200 µM acetylated fluorometric substrate
Reference: 10005019-25
€0.00 (tax incl.)
An HDAC inhibitor with an IC50 value of 30 µM when tested in HeLa cell nuclear extracts using 200 µM acetylated fluorometric substrate
Reference: 10005019-5
€0.00 (tax incl.)
An HDAC inhibitor with an IC50 value of 30 µM when tested in HeLa cell nuclear extracts using 200 µM acetylated fluorometric substrate
Reference: 10005031-100
€0.00 (tax incl.)
A relatively non-selective inhibitor of all NOS isoforms with Ki values 0.18, 0.4, and 6 µM for nNOs (rat), eNOS (human), and iNOS (mouse), respectively
Reference: 10005031-25
€0.00 (tax incl.)
A relatively non-selective inhibitor of all NOS isoforms with Ki values 0.18, 0.4, and 6 µM for nNOs (rat), eNOS (human), and iNOS (mouse), respectively
Reference: 10005031-5
€0.00 (tax incl.)
A relatively non-selective inhibitor of all NOS isoforms with Ki values 0.18, 0.4, and 6 µM for nNOs (rat), eNOS (human), and iNOS (mouse), respectively
Reference: 10005031-50
€0.00 (tax incl.)
A relatively non-selective inhibitor of all NOS isoforms with Ki values 0.18, 0.4, and 6 µM for nNOs (rat), eNOS (human), and iNOS (mouse), respectively
Reference: 10005033-10
€0.00 (tax incl.)
A selective antagonist of S1P binding to the S1P3 receptor; blocks calcium increase in HeLa cells by about 40% at 10 µM
Reference: 10005033-25
€0.00 (tax incl.)
A selective antagonist of S1P binding to the S1P3 receptor; blocks calcium increase in HeLa cells by about 40% at 10 µM
Reference: 10005033-5
€0.00 (tax incl.)
A selective antagonist of S1P binding to the S1P3 receptor; blocks calcium increase in HeLa cells by about 40% at 10 µM
Reference: 10005033-50
€0.00 (tax incl.)
A selective antagonist of S1P binding to the S1P3 receptor; blocks calcium increase in HeLa cells by about 40% at 10 µM
Reference: 10005067-1
€0.00 (tax incl.)
A selective inhibitor of the 20-HETE synthase, CYP4A11, exhibiting an IC50 values of 8.8 nM when tested in human renal microsomes
Reference: 10005067-10
€0.00 (tax incl.)
A selective inhibitor of the 20-HETE synthase, CYP4A11, exhibiting an IC50 values of 8.8 nM when tested in human renal microsomes
Reference: 10005067-5
€0.00 (tax incl.)
A selective inhibitor of the 20-HETE synthase, CYP4A11, exhibiting an IC50 values of 8.8 nM when tested in human renal microsomes
Reference: 10005067-50
€0.00 (tax incl.)
A selective inhibitor of the 20-HETE synthase, CYP4A11, exhibiting an IC50 values of 8.8 nM when tested in human renal microsomes
Reference: 10005072-1
€0.00 (tax incl.)
A labeled analog of AEA that is non-fluorescent when outside the cell but upon transport into the cell, is cleaved by esterases to give a bright fluorescence at 530 nm; used as an alternative substrate to study AEA...
Reference: 10005072-100
€0.00 (tax incl.)
A labeled analog of AEA that is non-fluorescent when outside the cell but upon transport into the cell, is cleaved by esterases to give a bright fluorescence at 530 nm; used as an alternative substrate to study AEA...
Reference: 10005072-500
€0.00 (tax incl.)
A labeled analog of AEA that is non-fluorescent when outside the cell but upon transport into the cell, is cleaved by esterases to give a bright fluorescence at 530 nm; used as an alternative substrate to study AEA...
Reference: 10005102-1
€0.00 (tax incl.)
A selective, potent inhibitor of rat FAAH (Ki = 0.57 nM); exhibited IC50 values of 0.81, 83 nM, and 50 µM for FAAH, TGH, and an uncharacterized hydrolase (KIAA1363), respectively, when screened against the serine...
Reference: 10005102-10
€0.00 (tax incl.)
A selective, potent inhibitor of rat FAAH (Ki = 0.57 nM); exhibited IC50 values of 0.81, 83 nM, and 50 µM for FAAH, TGH, and an uncharacterized hydrolase (KIAA1363), respectively, when screened against the serine...
Reference: 10005102-5
€0.00 (tax incl.)
A selective, potent inhibitor of rat FAAH (Ki = 0.57 nM); exhibited IC50 values of 0.81, 83 nM, and 50 µM for FAAH, TGH, and an uncharacterized hydrolase (KIAA1363), respectively, when screened against the serine...
Reference: 10005102-500
€0.00 (tax incl.)
A selective, potent inhibitor of rat FAAH (Ki = 0.57 nM); exhibited IC50 values of 0.81, 83 nM, and 50 µM for FAAH, TGH, and an uncharacterized hydrolase (KIAA1363), respectively, when screened against the serine...
Reference: 10005166-100
€0.00 (tax incl.)
An isoflavone; binds to ERβ (Ki = 2.8 µM) but not ERα up to 1 mM; estrogenic in vitro, increasing ERE-mediated gene transcription via ERβ (EC50 = 2.8 µM); an inhibitor of CAVII and CAXII (Kis = 4.2 and 56 nM,...
Reference: 10005166-1
€0.00 (tax incl.)
An isoflavone; binds to ERβ (Ki = 2.8 µM) but not ERα up to 1 mM; estrogenic in vitro, increasing ERE-mediated gene transcription via ERβ (EC50 = 2.8 µM); an inhibitor of CAVII and CAXII (Kis = 4.2 and 56 nM,...
Reference: 10005166-500
€0.00 (tax incl.)
An isoflavone; binds to ERβ (Ki = 2.8 µM) but not ERα up to 1 mM; estrogenic in vitro, increasing ERE-mediated gene transcription via ERβ (EC50 = 2.8 µM); an inhibitor of CAVII and CAXII (Kis = 4.2 and 56 nM,...
Reference: 10005166-5
€0.00 (tax incl.)
An isoflavone; binds to ERβ (Ki = 2.8 µM) but not ERα up to 1 mM; estrogenic in vitro, increasing ERE-mediated gene transcription via ERβ (EC50 = 2.8 µM); an inhibitor of CAVII and CAXII (Kis = 4.2 and 56 nM,...
Reference: 10005167-100
€0.00 (tax incl.)
An isoflavonoid phytoestrogen with kinase inhibitory, anticancer, pro-cancer, hepatoprotective, and antiviral properties; inhibits EGFR, pp50v-Src, and pp110gag-fes (IC50s = 6, 7-8, and 6.5 µg/ml, respectively);...
Reference: 10005167-1
€0.00 (tax incl.)
An isoflavonoid phytoestrogen with kinase inhibitory, anticancer, pro-cancer, hepatoprotective, and antiviral properties; inhibits EGFR, pp50v-Src, and pp110gag-fes (IC50s = 6, 7-8, and 6.5 µg/ml, respectively);...
Reference: 10005167-250
€0.00 (tax incl.)
An isoflavonoid phytoestrogen with kinase inhibitory, anticancer, pro-cancer, hepatoprotective, and antiviral properties; inhibits EGFR, pp50v-Src, and pp110gag-fes (IC50s = 6, 7-8, and 6.5 µg/ml, respectively);...
Reference: 10005167-500
€0.00 (tax incl.)
An isoflavonoid phytoestrogen with kinase inhibitory, anticancer, pro-cancer, hepatoprotective, and antiviral properties; inhibits EGFR, pp50v-Src, and pp110gag-fes (IC50s = 6, 7-8, and 6.5 µg/ml, respectively);...
Reference: 10005169-10
€0.00 (tax incl.)
A flavonoid; reduces autophagy, decreases the levels of ROS and MDA content, and increases total antioxidant capacity in the kidney in a mouse model of cadmium-induced autophagy at 5-100 mg/kg; reduces tumor growth in...
Reference: 10005169-100
€0.00 (tax incl.)
A flavonoid; reduces autophagy, decreases the levels of ROS and MDA content, and increases total antioxidant capacity in the kidney in a mouse model of cadmium-induced autophagy at 5-100 mg/kg; reduces tumor growth in...
Reference: 10005169-5
€0.00 (tax incl.)
A flavonoid; reduces autophagy, decreases the levels of ROS and MDA content, and increases total antioxidant capacity in the kidney in a mouse model of cadmium-induced autophagy at 5-100 mg/kg; reduces tumor growth in...
Reference: 10005169-50
€0.00 (tax incl.)
A flavonoid; reduces autophagy, decreases the levels of ROS and MDA content, and increases total antioxidant capacity in the kidney in a mouse model of cadmium-induced autophagy at 5-100 mg/kg; reduces tumor growth in...
Reference: 10005174-1
€0.00 (tax incl.)
A lignan with diverse biological activities; reduces LPS-induced production of NO and PGE2 in RAW 264.7 cells; cytotoxic to colon 26 cancer cells (LC50 = 9 µg/ml); increases the lifespan of C. elegans at 100 µM;...
Reference: 10005174-10
€0.00 (tax incl.)
A lignan with diverse biological activities; reduces LPS-induced production of NO and PGE2 in RAW 264.7 cells; cytotoxic to colon 26 cancer cells (LC50 = 9 µg/ml); increases the lifespan of C. elegans at 100 µM;...
Reference: 10005174-25
€0.00 (tax incl.)
A lignan with diverse biological activities; reduces LPS-induced production of NO and PGE2 in RAW 264.7 cells; cytotoxic to colon 26 cancer cells (LC50 = 9 µg/ml); increases the lifespan of C. elegans at 100 µM;...
Reference: 10005174-5
€0.00 (tax incl.)
A lignan with diverse biological activities; reduces LPS-induced production of NO and PGE2 in RAW 264.7 cells; cytotoxic to colon 26 cancer cells (LC50 = 9 µg/ml); increases the lifespan of C. elegans at 100 µM;...
Reference: 10005186-10
€0.00 (tax incl.)
A potent antagonist for the human IP (prostacyclin) receptor that antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cAMP accumulation in a dose-dependent manner;...
Reference: 10005186-25
€0.00 (tax incl.)
A potent antagonist for the human IP (prostacyclin) receptor that antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cAMP accumulation in a dose-dependent manner;...
Reference: 10005186-5
€0.00 (tax incl.)
A potent antagonist for the human IP (prostacyclin) receptor that antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cAMP accumulation in a dose-dependent manner;...
Reference: 10005186-50
€0.00 (tax incl.)
A potent antagonist for the human IP (prostacyclin) receptor that antagonizes the carbaprostacyclin-induced activation of human neuroblastoma adenylate cyclase, blocking cAMP accumulation in a dose-dependent manner;...
Reference: 10005189-1
€0.00 (tax incl.)
Suppresses both constitutive and hypoxia-induced levels of HIF-1α in cancer cells, resulting in reduced expression of HIF-1α target genes; increases chemo- or radiosensitivity of tumors
Reference: 10005189-10
€0.00 (tax incl.)
Suppresses both constitutive and hypoxia-induced levels of HIF-1α in cancer cells, resulting in reduced expression of HIF-1α target genes; increases chemo- or radiosensitivity of tumors
Reference: 10005189-25
€0.00 (tax incl.)
Suppresses both constitutive and hypoxia-induced levels of HIF-1α in cancer cells, resulting in reduced expression of HIF-1α target genes; increases chemo- or radiosensitivity of tumors
Reference: 10005189-5
€0.00 (tax incl.)
Suppresses both constitutive and hypoxia-induced levels of HIF-1α in cancer cells, resulting in reduced expression of HIF-1α target genes; increases chemo- or radiosensitivity of tumors
Reference: 10005229-10
€0.00 (tax incl.)
A proapoptoic compound with selectivity for cancer cells; induces apoptosis in vitro in various cancer cell lines (IC50 = 0.89-2.69 µM)
Reference: 10005229-5
€0.00 (tax incl.)
A proapoptoic compound with selectivity for cancer cells; induces apoptosis in vitro in various cancer cell lines (IC50 = 0.89-2.69 µM)
Reference: 10005229-50
€0.00 (tax incl.)
A proapoptoic compound with selectivity for cancer cells; induces apoptosis in vitro in various cancer cell lines (IC50 = 0.89-2.69 µM)
Reference: 10005254-1
€0.00 (tax incl.)
A melatonin metabolite first identified in rat brain that has antioxidant and free radical scavenging activities in several experimental models; may be measured in plasma as an index of melatonin synthesis and...
Reference: 10005254-10
€0.00 (tax incl.)
A melatonin metabolite first identified in rat brain that has antioxidant and free radical scavenging activities in several experimental models; may be measured in plasma as an index of melatonin synthesis and...
Reference: 10005254-5
€0.00 (tax incl.)
A melatonin metabolite first identified in rat brain that has antioxidant and free radical scavenging activities in several experimental models; may be measured in plasma as an index of melatonin synthesis and...
Reference: 10005254-50
€0.00 (tax incl.)
A melatonin metabolite first identified in rat brain that has antioxidant and free radical scavenging activities in several experimental models; may be measured in plasma as an index of melatonin synthesis and...
Reference: 10005263-10
€0.00 (tax incl.)
An inhibitor of fatty acid synthesis that blocks the synthesis of malonyl-CoA by acetyl-CoA carboxylase (ACC)
Reference: 10005263-100
€0.00 (tax incl.)
An inhibitor of fatty acid synthesis that blocks the synthesis of malonyl-CoA by acetyl-CoA carboxylase (ACC)
Reference: 10005263-5
€0.00 (tax incl.)
An inhibitor of fatty acid synthesis that blocks the synthesis of malonyl-CoA by acetyl-CoA carboxylase (ACC)
Reference: 10005263-50
€0.00 (tax incl.)
An inhibitor of fatty acid synthesis that blocks the synthesis of malonyl-CoA by acetyl-CoA carboxylase (ACC)
Reference: 10005270-1
€0.00 (tax incl.)
A stable inhibitor of FASN that leads to profound weight loss and feeding inhibition in both high-fat diet wild type obese and leptin-deficient ob/ob mice
Reference: 10005270-10
€0.00 (tax incl.)
A stable inhibitor of FASN that leads to profound weight loss and feeding inhibition in both high-fat diet wild type obese and leptin-deficient ob/ob mice
Reference: 10005270-5
€0.00 (tax incl.)
A stable inhibitor of FASN that leads to profound weight loss and feeding inhibition in both high-fat diet wild type obese and leptin-deficient ob/ob mice
Reference: 10005276-10
€0.00 (tax incl.)
A PDMP mixture containing D-threo (1R,2R) and L-threo (1S,2S) PDMP; inhibits glucosylceramide synthase by 33 and 48% in MDCK cell homogenates at 5 and 10 µM; reduces the synthesis of glucosylceramide increases...
Reference: 10005276-100
€0.00 (tax incl.)
A PDMP mixture containing D-threo (1R,2R) and L-threo (1S,2S) PDMP; inhibits glucosylceramide synthase by 33 and 48% in MDCK cell homogenates at 5 and 10 µM; reduces the synthesis of glucosylceramide increases...
Reference: 10005276-5
€0.00 (tax incl.)
A PDMP mixture containing D-threo (1R,2R) and L-threo (1S,2S) PDMP; inhibits glucosylceramide synthase by 33 and 48% in MDCK cell homogenates at 5 and 10 µM; reduces the synthesis of glucosylceramide increases...
Reference: 10005276-50
€0.00 (tax incl.)
A PDMP mixture containing D-threo (1R,2R) and L-threo (1S,2S) PDMP; inhibits glucosylceramide synthase by 33 and 48% in MDCK cell homogenates at 5 and 10 µM; reduces the synthesis of glucosylceramide increases...
Reference: 10005278-1
€0.00 (tax incl.)
An enhancer of sphingolipid biosynthesis; increases glucosylceramide synthase activity by 4 and 8% when used at concentrations of 5 and 2.5 µM, respectively, in an enzyme assay; increases the activity of ganglioside...
Reference: 10005278-10
€0.00 (tax incl.)
An enhancer of sphingolipid biosynthesis; increases glucosylceramide synthase activity by 4 and 8% when used at concentrations of 5 and 2.5 µM, respectively, in an enzyme assay; increases the activity of ganglioside...
Reference: 10005278-5
€0.00 (tax incl.)
An enhancer of sphingolipid biosynthesis; increases glucosylceramide synthase activity by 4 and 8% when used at concentrations of 5 and 2.5 µM, respectively, in an enzyme assay; increases the activity of ganglioside...
Reference: 10005291-1
€0.00 (tax incl.)
Contains PRIMA-1, p53 (Phospho-Ser392) Polyclonal Antibody, (±)-Nutlin-3, and Caylin-2
Reference: 10005368-1
€0.00 (tax incl.)
A PPARα agonist (EC50s = 18 and 30 μM for mouse and human receptors, respectively, in a transactivation assay); selective for PPARα over PPARγ (EC50s = 300 and 200 μM for mouse and human receptors, respectively) and...
Reference: 10005368-10
€0.00 (tax incl.)
A PPARα agonist (EC50s = 18 and 30 μM for mouse and human receptors, respectively, in a transactivation assay); selective for PPARα over PPARγ (EC50s = 300 and 200 μM for mouse and human receptors, respectively) and...
Reference: 10005368-5
€0.00 (tax incl.)
A PPARα agonist (EC50s = 18 and 30 μM for mouse and human receptors, respectively, in a transactivation assay); selective for PPARα over PPARγ (EC50s = 300 and 200 μM for mouse and human receptors, respectively) and...
Reference: 10005368-50
€0.00 (tax incl.)
A PPARα agonist (EC50s = 18 and 30 μM for mouse and human receptors, respectively, in a transactivation assay); selective for PPARα over PPARγ (EC50s = 300 and 200 μM for mouse and human receptors, respectively) and...
Reference: 10005426-100
€0.00 (tax incl.)
An anti-obesity drug that inhibits gastric, pancreatic, and carboxyl ester lipases, preventing hydrolysis of triglycerides to free fatty acids and monoglycerides; potently inhibits human recombinant DAGLα (IC50 = 60...
Reference: 10005426-250
€0.00 (tax incl.)
An anti-obesity drug that inhibits gastric, pancreatic, and carboxyl ester lipases, preventing hydrolysis of triglycerides to free fatty acids and monoglycerides; potently inhibits human recombinant DAGLα (IC50 = 60...
Reference: 10005426-50
€0.00 (tax incl.)
An anti-obesity drug that inhibits gastric, pancreatic, and carboxyl ester lipases, preventing hydrolysis of triglycerides to free fatty acids and monoglycerides; potently inhibits human recombinant DAGLα (IC50 = 60...
Reference: 10005426-500
€0.00 (tax incl.)
An anti-obesity drug that inhibits gastric, pancreatic, and carboxyl ester lipases, preventing hydrolysis of triglycerides to free fatty acids and monoglycerides; potently inhibits human recombinant DAGLα (IC50 = 60...

DDA

Reference: 10005432-10
€0.00 (tax incl.)
A prominent member of a class of reactive LO-catalyzed peroxidative decomposition products of unsaturated fatty acids that are formed when diatoms are crushed or eaten

DDA

Reference: 10005432-25
€0.00 (tax incl.)
A prominent member of a class of reactive LO-catalyzed peroxidative decomposition products of unsaturated fatty acids that are formed when diatoms are crushed or eaten

DDA

Reference: 10005432-5
€0.00 (tax incl.)
A prominent member of a class of reactive LO-catalyzed peroxidative decomposition products of unsaturated fatty acids that are formed when diatoms are crushed or eaten

DDA

Reference: 10005432-50
€0.00 (tax incl.)
A prominent member of a class of reactive LO-catalyzed peroxidative decomposition products of unsaturated fatty acids that are formed when diatoms are crushed or eaten
Reference: 10005537-1
€0.00 (tax incl.)
An arachidonoyl amino acid; an activator of TRPV1 and TRPV4 (EC50s = 28 and 21 µM, respectively); increases calcium flux in HIT-T15 pancreatic β-cells and INS-1 rat islet cells at 10 µM; increases insulin secretion...
Reference: 10005537-10
€0.00 (tax incl.)
An arachidonoyl amino acid; an activator of TRPV1 and TRPV4 (EC50s = 28 and 21 µM, respectively); increases calcium flux in HIT-T15 pancreatic β-cells and INS-1 rat islet cells at 10 µM; increases insulin secretion...
Reference: 10005537-5
€0.00 (tax incl.)
An arachidonoyl amino acid; an activator of TRPV1 and TRPV4 (EC50s = 28 and 21 µM, respectively); increases calcium flux in HIT-T15 pancreatic β-cells and INS-1 rat islet cells at 10 µM; increases insulin secretion...
Reference: 10005537-500
€0.00 (tax incl.)
An arachidonoyl amino acid; an activator of TRPV1 and TRPV4 (EC50s = 28 and 21 µM, respectively); increases calcium flux in HIT-T15 pancreatic β-cells and INS-1 rat islet cells at 10 µM; increases insulin secretion...
Reference: 10005583-1
€0.00 (tax incl.)
A potent, ATP-competitive inhibitor of ROCKs including p160ROCK (Ki = 140 nM) and ROCK-II (IC50 = 800 nM); also inhibits PRK2 with an IC50 value of 600 nM
Reference: 10005583-10
€0.00 (tax incl.)
A potent, ATP-competitive inhibitor of ROCKs including p160ROCK (Ki = 140 nM) and ROCK-II (IC50 = 800 nM); also inhibits PRK2 with an IC50 value of 600 nM
Reference: 10005583-5
€0.00 (tax incl.)
A potent, ATP-competitive inhibitor of ROCKs including p160ROCK (Ki = 140 nM) and ROCK-II (IC50 = 800 nM); also inhibits PRK2 with an IC50 value of 600 nM
Reference: 10005583-50
€0.00 (tax incl.)
A potent, ATP-competitive inhibitor of ROCKs including p160ROCK (Ki = 140 nM) and ROCK-II (IC50 = 800 nM); also inhibits PRK2 with an IC50 value of 600 nM

Menu

Settings