RA375

Tax included
RA375 is a RPN13 (26S proteasome regulatory subunit) inhibitor. RA375 activates UPR signaling, ROS production and apoptosis. RA375 exhibits ten-fold greater activity against cancer lines than RA190, reflecting its nitro ring substituents and the addition of a chloroacetamide warhead.
HY-136563

Data sheet

Size
Multiple sizes
Reactivity
Proteasome; Apoptosis; Reactive Oxygen Species
Application
Cancer-Kinase/protease